Drug discovery open innovation – beyond the Rule of 5.
Do you have a novel cell-based assay? Looking to find novel compounds custom designed to penetrate cells?
Our partner is offering access to a compound set designed with specific biological properties, using their many years of Pharma medicinal chemistry.
This particular set uses its amphiphilic design to enhance lipophilicity, and thus membrane permeability and cellular assay potency, whilst limiting potential metabolic liabilities.
It is currently a small collection with wide diversity built around the enhanced cellular absorption properties. We are providing the collection blind of structures, which would be revealed for hit compounds of interest. Our partner is interested in sharing access to their collection in return for an offer to use their design algorithm to assist in the selection and synthesis of hit related compounds.
Enhance your potential of success from cellular assays – contact us to discuss further.